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pukhtun

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D1 Antagonists= Zotepine

D2 Antagonism=Amisulpiride, Clozapine, sulpiride, thioridazine, Thioxanthines, Zotepine. Quetiapine

D3 Antagonism= Amisulpiride, Ziprasidone, Zotepine

D4 Antagonism= Clozapine, Ziprasidone, Zotepine.Olanzapine

[ch945] 1 Antagonism= Clozapine,Nefazadone, trazodone

[ch945] 2 Antagonism=mirtazapine, trazodone,yohimbine ( erectile dysfunction)

presynaptic [ch945] 2 agonism = clonidine, Lofexidine

Anti muscarinic= Chlorpromazine, Promazine, Thioridazine, periyclizine, Ziprasidone ( poor)

Anti cholinergic= Clozapine, Olanzapine, Quetiapine , delirium

Anti histaminic= Clozapine, Olanzapine, Ziprasidone, Zotepine.mirtazapine, trazodone

Weak D1 and D2 affinity= Clozapine

5HT1A antagonist= pindolol

Partial 5HT1A agonist= Buspirone

5HT2A antagonist= Risperidone, Aripiprazole, Zotepine. Weak Quetiapine, Ziprasidone, mirtazapine,Trazodone

5HT2A partial agonist= LSD

5HT2c antagonist= trazodone

5HT3= mirtazapine

SNRI= Duloxetine,venlafaxine, milnacipran, Amoxapine (with dopamine antagonist properties)

NARI= Reboxetine, Atomoxetine

Short acting opioid mu antagonist = Naloxone

Long acting opioid mu antagonist= Naltrexone

Non competitive NMDA antagonists= Phencyclidine, Ketamine.

Acetyl cholinesterase inhibitor= Donepazil and Galantamine

Acetyl and butyl cholinesterase inhibitors= Rivastigmine

Nictotinic agonistic= Gallantamine

NMDA block= Memantine

Methylphenidate and dextroamphetamines= Indirectly acting sympathomimmetics, weak inhibitors of catecholamine reuptake and inhibitors of MAO

Atomoxetine= Tricyclic like-phenylpropanolamine derivative

Beta adrenergic antagonist= Propanolol

Phosphodiesterase inhibitor= sildenafil (Viagra)

Side effects

[ch945] 2 blockade= agitation, impotence

[ch945] 1 Blockade= postural hypotension, anorgasmia, priapism, retrograde ejaculation.

D2 blockade= akathesia, EPSE, Hyperprolactenimea

5HT2A stimulation= agitation, akathesia, appetite loss, anorgasmia, impotence, reduce libido.Hyperthermia

5HT2c stimulation= agitation, hyperthermia, anorgasmia, impotence

5HT2c antagonism= weight gain

5HT1D stimulation= induce obsessions

5HT2A antagonism= reduces akathesia, reduces EPSE, slow wave sleep, anti depressant action

5HT1A stimulation= Reduces OCD, anti depressant action

5HT1A stimulation= Hyperprolactinaemia

Anti histamine= increase appetite, weight gain

5HT3 stimulation= GI discomfort, nausea, vomiting

Anticholinergic= Amnesia, delirium

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